TAE-684 KINOMEscan - Dataset (ID:20199)

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Small Molecule Protein Kd Conc unit
NVP-TAE684 MARK1 31.0
nM
NVP-TAE684 KCC4 30.0
nM
NVP-TAE684 PAK3 29.0
nM
NVP-TAE684 ACVR1 29.0
nM
NVP-TAE684 FRK 27.0
nM
NVP-TAE684 AMPK-alpha1 27.0
nM
NVP-TAE684 RSK4(Kin.Dom.1-N-terminal) 27.0
nM
NVP-TAE684 KIT(D816V) 26.0
nM
NVP-TAE684 TAOK1 25.0
nM
NVP-TAE684 TSSK1 25.0
nM
NVP-TAE684 YANK2 24.0
nM
NVP-TAE684 YES 23.0
nM
NVP-TAE684 BTK 23.0
nM
NVP-TAE684 SBK1 21.0
nM
NVP-TAE684 SLK 21.0
nM
NVP-TAE684 PLK1 20.0
nM
NVP-TAE684 ABL1(F317L)-phosphorylated 19.0
nM
NVP-TAE684 MERTK 19.0
nM
NVP-TAE684 JAK3(JH1domain-catalytic) 17.0
nM
NVP-TAE684 RSK2(Kin.Dom.1-N-terminal) 17.0
nM
NVP-TAE684 PHKG1 17.0
nM
NVP-TAE684 SIK2 17.0
nM
NVP-TAE684 DCAMKL2 16.0
nM
NVP-TAE684 JAK2(JH1domain-catalytic) 16.0
nM
NVP-TAE684 TIE1 15.0
nM