TAE-684 KINOMEscan - Dataset (ID:20199)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
NVP-TAE684 | MARK1 | 31.0 | nM |
NVP-TAE684 | KCC4 | 30.0 | nM |
NVP-TAE684 | PAK3 | 29.0 | nM |
NVP-TAE684 | ACVR1 | 29.0 | nM |
NVP-TAE684 | FRK | 27.0 | nM |
NVP-TAE684 | AMPK-alpha1 | 27.0 | nM |
NVP-TAE684 | RSK4(Kin.Dom.1-N-terminal) | 27.0 | nM |
NVP-TAE684 | KIT(D816V) | 26.0 | nM |
NVP-TAE684 | TAOK1 | 25.0 | nM |
NVP-TAE684 | TSSK1 | 25.0 | nM |
NVP-TAE684 | YANK2 | 24.0 | nM |
NVP-TAE684 | YES | 23.0 | nM |
NVP-TAE684 | BTK | 23.0 | nM |
NVP-TAE684 | SBK1 | 21.0 | nM |
NVP-TAE684 | SLK | 21.0 | nM |
NVP-TAE684 | PLK1 | 20.0 | nM |
NVP-TAE684 | ABL1(F317L)-phosphorylated | 19.0 | nM |
NVP-TAE684 | MERTK | 19.0 | nM |
NVP-TAE684 | JAK3(JH1domain-catalytic) | 17.0 | nM |
NVP-TAE684 | RSK2(Kin.Dom.1-N-terminal) | 17.0 | nM |
NVP-TAE684 | PHKG1 | 17.0 | nM |
NVP-TAE684 | SIK2 | 17.0 | nM |
NVP-TAE684 | DCAMKL2 | 16.0 | nM |
NVP-TAE684 | JAK2(JH1domain-catalytic) | 16.0 | nM |
NVP-TAE684 | TIE1 | 15.0 | nM |