TAE-684 KINOMEscan - Dataset (ID:20199)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
NVP-TAE684 | TTK | 50.0 | nM |
NVP-TAE684 | AMPK-alpha2 | 49.0 | nM |
NVP-TAE684 | LCK | 49.0 | nM |
NVP-TAE684 | KIT(L576P) | 49.0 | nM |
NVP-TAE684 | CSF1R | 48.0 | nM |
NVP-TAE684 | ERK5 | 48.0 | nM |
NVP-TAE684 | OSR1 | 48.0 | nM |
NVP-TAE684 | FGFR1 | 47.0 | nM |
NVP-TAE684 | EGFR(L858R) | 46.0 | nM |
NVP-TAE684 | TIE2 | 46.0 | nM |
NVP-TAE684 | IRAK1 | 45.0 | nM |
NVP-TAE684 | TAOK3 | 44.0 | nM |
NVP-TAE684 | AURKA | 44.0 | nM |
NVP-TAE684 | MARK2 | 44.0 | nM |
NVP-TAE684 | MKNK2 | 44.0 | nM |
NVP-TAE684 | CHEK1 | 44.0 | nM |
NVP-TAE684 | M3K12 | 42.0 | nM |
NVP-TAE684 | EPHA1 | 39.0 | nM |
NVP-TAE684 | ABL1(Q252H)-nonphosphorylated | 39.0 | nM |
NVP-TAE684 | ROCK1 | 37.0 | nM |
NVP-TAE684 | PTK6 | 36.0 | nM |
NVP-TAE684 | ITK | 34.0 | nM |
NVP-TAE684 | FLT3(R834Q) | 34.0 | nM |
NVP-TAE684 | RSK3(Kin.Dom.1-N-terminal) | 33.0 | nM |
NVP-TAE684 | AURKC | 33.0 | nM |