TAE-684 KINOMEscan - Dataset (ID:20199)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
NVP-TAE684 | LOK | 82.0 | nM |
NVP-TAE684 | CLK2 | 82.0 | nM |
NVP-TAE684 | MYO3B | 81.0 | nM |
NVP-TAE684 | EGFR(E746-A750del) | 81.0 | nM |
NVP-TAE684 | KIT(V559D) | 81.0 | nM |
NVP-TAE684 | KPCD1 | 80.0 | nM |
NVP-TAE684 | EGFR(L747-T751del,Sins) | 79.0 | nM |
NVP-TAE684 | TYK2(JH1domain-catalytic) | 77.0 | nM |
NVP-TAE684 | IRAK4 | 77.0 | nM |
NVP-TAE684 | ABL1(H396P)-nonphosphorylated | 73.0 | nM |
NVP-TAE684 | CHK2 | 72.0 | nM |
NVP-TAE684 | EGFR(L747-E749del, A750P) | 72.0 | nM |
NVP-TAE684 | ABL1(Q252H)-phosphorylated | 70.0 | nM |
NVP-TAE684 | MYO3A | 67.0 | nM |
NVP-TAE684 | JNK3 | 67.0 | nM |
NVP-TAE684 | M4K3 | 65.0 | nM |
NVP-TAE684 | MET(M1250T) | 64.0 | nM |
NVP-TAE684 | M3K13 | 57.0 | nM |
NVP-TAE684 | RIPK5 | 57.0 | nM |
NVP-TAE684 | ACVRL1 | 57.0 | nM |
NVP-TAE684 | YANK3 | 55.0 | nM |
NVP-TAE684 | ABL1(F317L)-nonphosphorylated | 54.0 | nM |
NVP-TAE684 | SgK110 | 54.0 | nM |
NVP-TAE684 | ABL1(T315I)-nonphosphorylated | 52.0 | nM |
NVP-TAE684 | KKCC1 | 50.0 | nM |