TAE-684 KINOMEscan - Dataset (ID:20199)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| NVP-TAE684 | KIT | 110.0 | nM |
| NVP-TAE684 | KIT(A829P) | 220.0 | nM |
| NVP-TAE684 | KIT(D816H) | 140.0 | nM |
| NVP-TAE684 | KIT(D816V) | 26.0 | nM |
| NVP-TAE684 | KIT(L576P) | 49.0 | nM |
| NVP-TAE684 | KIT(V559D) | 81.0 | nM |
| NVP-TAE684 | KIT(V559D,T670I) | 130.0 | nM |
| NVP-TAE684 | KIT(V559D,V654A) | 1200.0 | nM |
| NVP-TAE684 | LATS1 | 1600.0 | nM |
| NVP-TAE684 | LATS2 | 2000.0 | nM |
| NVP-TAE684 | LCK | 49.0 | nM |
| NVP-TAE684 | LIMK1 | 1100.0 | nM |
| NVP-TAE684 | LIMK2 | 1100.0 | nM |
| NVP-TAE684 | LKB1 | nM | |
| NVP-TAE684 | LOK | 82.0 | nM |
| NVP-TAE684 | LRRK2 | 1.4 | nM |
| NVP-TAE684 | LRRK2(G2019S) | 0.9 | nM |
| NVP-TAE684 | LTK | 1.0 | nM |
| NVP-TAE684 | LYN | 280.0 | nM |
| NVP-TAE684 | M3K13 | 57.0 | nM |
| NVP-TAE684 | MAK | nM | |
| NVP-TAE684 | MAP3K1 | 4300.0 | nM |
| NVP-TAE684 | MAP3K15 | 800.0 | nM |
| NVP-TAE684 | M3K2 | 110.0 | nM |
| NVP-TAE684 | MAP3K3 | 320.0 | nM |