TAE-684 KINOMEscan - Dataset (ID:20199)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| NVP-TAE684 | FES | 4.8 | nM |
| NVP-TAE684 | FGFR1 | 47.0 | nM |
| NVP-TAE684 | FGFR2 | 250.0 | nM |
| NVP-TAE684 | FGFR3 | 95.0 | nM |
| NVP-TAE684 | FGFR3(G697C) | 120.0 | nM |
| NVP-TAE684 | FGFR4 | 110.0 | nM |
| NVP-TAE684 | FGR | 120.0 | nM |
| NVP-TAE684 | VGFR1 | 550.0 | nM |
| NVP-TAE684 | FLT3 | 15.0 | nM |
| NVP-TAE684 | FLT3(D835H) | 4.9 | nM |
| NVP-TAE684 | FLT3(D835Y) | 2.0 | nM |
| NVP-TAE684 | FLT3(ITD) | 8.6 | nM |
| NVP-TAE684 | FLT3(K663Q) | 8.2 | nM |
| NVP-TAE684 | FLT3(N841I) | 11.0 | nM |
| NVP-TAE684 | FLT3(R834Q) | 34.0 | nM |
| NVP-TAE684 | FLT4 | 170.0 | nM |
| NVP-TAE684 | FRK | 27.0 | nM |
| NVP-TAE684 | FYN | 1400.0 | nM |
| NVP-TAE684 | GAK | 5.3 | nM |
| NVP-TAE684 | GCN2(Kin.Dom.2,S808G) | 1100.0 | nM |
| NVP-TAE684 | GRK1 | 410.0 | nM |
| NVP-TAE684 | GRK4 | 3500.0 | nM |
| NVP-TAE684 | GRK7 | 360.0 | nM |
| NVP-TAE684 | GSK3A | nM | |
| NVP-TAE684 | GSK3B | nM |