Imatinib KINOMEscan - Dataset (ID:20198)

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Small Molecule Protein Kd Conc unit
Imatinib TYK2(JH2domain-pseudokinase) 8700.0
nM
Imatinib PLK4 7800.0
nM
Imatinib EGFR(L747-E749del, A750P) 7600.0
nM
Imatinib FLT3(ITD) 6300.0
nM
Imatinib CDK11 5500.0
nM
Imatinib DRAK1 5300.0
nM
Imatinib JNK1 5000.0
nM
Imatinib CLK1 4500.0
nM
Imatinib TNNI3K 4300.0
nM
Imatinib BRAF(V600E) 3300.0
nM
Imatinib FYN 3100.0
nM
Imatinib JNK3 3100.0
nM
Imatinib MLTK 2600.0
nM
Imatinib KIT(V559D,T670I) 2500.0
nM
Imatinib FGR 2400.0
nM
Imatinib CLK4 2100.0
nM
Imatinib MELK 1900.0
nM
Imatinib RAF1 1700.0
nM
Imatinib FRK 1500.0
nM
Imatinib EPHA8 1400.0
nM
Imatinib IRAK1 1200.0
nM
Imatinib GAK 1000.0
nM
Imatinib KIT(D816V) 980.0
nM
Imatinib HIPK4 960.0
nM
Imatinib LYN 890.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records