Imatinib KINOMEscan - Dataset (ID:20198)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Imatinib | DDR1 | 0.7 | nM |
Imatinib | ABL1-nonphosphorylated | 1.1 | nM |
Imatinib | ABL1(Q252H)-nonphosphorylated | 1.8 | nM |
Imatinib | ABL1(F317L)-nonphosphorylated | 2.5 | nM |
Imatinib | ABL1(H396P)-nonphosphorylated | 5.9 | nM |
Imatinib | ABL1(F317I)-nonphosphorylated | 8.3 | nM |
Imatinib | ABL2 | 10.0 | nM |
Imatinib | CSF1R | 11.0 | nM |
Imatinib | KIT | 13.0 | nM |
Imatinib | KIT(L576P) | 14.0 | nM |
Imatinib | PGFRB | 14.0 | nM |
Imatinib | KIT(A829P) | 15.0 | nM |
Imatinib | DDR2 | 15.0 | nM |
Imatinib | KIT(V559D) | 15.0 | nM |
Imatinib | ABL1-phosphorylated | 21.0 | nM |
Imatinib | PGFRA | 31.0 | nM |
Imatinib | LCK | 40.0 | nM |
Imatinib | ABL1(M351T)-phosphorylated | 44.0 | nM |
Imatinib | ABL1(H396P)-phosphorylated | 65.0 | nM |
Imatinib | KIT(V559D,V654A) | 91.0 | nM |
Imatinib | ABL1(Q252H)-phosphorylated | 92.0 | nM |
Imatinib | ABL1(F317L)-phosphorylated | 110.0 | nM |
Imatinib | ABL1(Y253F)-phosphorylated | 130.0 | nM |
Imatinib | ABL1(E255K)-phosphorylated | 170.0 | nM |
Imatinib | PI42C | 380.0 | nM |