VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Tozasertib | FES | 7400.0 | nM |
| Tozasertib | FGFR1 | 550.0 | nM |
| Tozasertib | FGFR2 | 570.0 | nM |
| Tozasertib | FGFR3 | 860.0 | nM |
| Tozasertib | FGFR3(G697C) | 820.0 | nM |
| Tozasertib | FGFR4 | 7200.0 | nM |
| Tozasertib | FGR | 790.0 | nM |
| Tozasertib | VGFR1 | 100.0 | nM |
| Tozasertib | FLT3 | 6.5 | nM |
| Tozasertib | FLT3(D835H) | 14.0 | nM |
| Tozasertib | FLT3(D835Y) | 55.0 | nM |
| Tozasertib | FLT3(ITD) | 45.0 | nM |
| Tozasertib | FLT3(K663Q) | 4.8 | nM |
| Tozasertib | FLT3(N841I) | 4.3 | nM |
| Tozasertib | FLT3(R834Q) | 130.0 | nM |
| Tozasertib | FLT4 | 1900.0 | nM |
| Tozasertib | FRK | 3800.0 | nM |
| Tozasertib | FYN | 530.0 | nM |
| Tozasertib | GAK | 3200.0 | nM |
| Tozasertib | GCN2(Kin.Dom.2,S808G) | 1900.0 | nM |
| Tozasertib | GRK1 | nM | |
| Tozasertib | GRK4 | 400.0 | nM |
| Tozasertib | GRK7 | nM | |
| Tozasertib | GSK3A | nM | |
| Tozasertib | GSK3B | nM |