VX-680 KINOMEscan - Dataset (ID:20197)

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Small Molecule Protein Kd Conc unit
Tozasertib AKT2
nM
Tozasertib AKT3
nM
Tozasertib ALK 3100.0
nM
Tozasertib AMPK-alpha1 1100.0
nM
Tozasertib AMPK-alpha2 350.0
nM
Tozasertib ANKK1 5600.0
nM
Tozasertib AURKA 3.9
nM
Tozasertib AURKB 7.4
nM
Tozasertib AURKC 6.3
nM
Tozasertib AXL 210.0
nM
Tozasertib BIKE 65.0
nM
Tozasertib BLK 2200.0
nM
Tozasertib BMPR1A
nM
Tozasertib BMPR1B 1100.0
nM
Tozasertib BMPR2 7100.0
nM
Tozasertib BMX 2600.0
nM
Tozasertib BRAF
nM
Tozasertib BRAF(V600E)
nM
Tozasertib BRSK1 8400.0
nM
Tozasertib BRSK2
nM
Tozasertib BTK 4400.0
nM
Tozasertib CAMK1 7000.0
nM
Tozasertib CAMK1D 4900.0
nM
Tozasertib CAMK1G 6500.0
nM
Tozasertib CAMK2A
nM