VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Tozasertib | RET | 28.0 | nM |
| Tozasertib | DDR1 | 28.0 | nM |
| Tozasertib | EPHB6 | 28.0 | nM |
| Tozasertib | TRKA | 38.0 | nM |
| Tozasertib | MYLK2 | 43.0 | nM |
| Tozasertib | FLT3(ITD) | 45.0 | nM |
| Tozasertib | CDKL2 | 49.0 | nM |
| Tozasertib | YSK4 | 51.0 | nM |
| Tozasertib | FLT3(D835Y) | 55.0 | nM |
| Tozasertib | LCK | 61.0 | nM |
| Tozasertib | BIKE | 65.0 | nM |
| Tozasertib | M4K1 | 72.0 | nM |
| Tozasertib | TAOK3 | 81.0 | nM |
| Tozasertib | SRPK1 | 82.0 | nM |
| Tozasertib | SLK | 82.0 | nM |
| Tozasertib | TNK1 | 83.0 | nM |
| Tozasertib | MAP4K5 | 83.0 | nM |
| Tozasertib | VGFR1 | 100.0 | nM |
| Tozasertib | LOK | 120.0 | nM |
| Tozasertib | PIP5K1A | 130.0 | nM |
| Tozasertib | FLT3(R834Q) | 130.0 | nM |
| Tozasertib | PIP5K2B | 140.0 | nM |
| Tozasertib | SRC | 170.0 | nM |
| Tozasertib | M3K13 | 180.0 | nM |
| Tozasertib | M3K12 | 190.0 | nM |