HKI-272 KINOMEscan-2 - Dataset (ID:20195)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Neratinib | KIT(V559D) | nM | |
Neratinib | KIT(V559D,T670I) | nM | |
Neratinib | KIT(V559D,V654A) | nM | |
Neratinib | KKCC1 | nM | |
Neratinib | KPCD | nM | |
Neratinib | KPCD1 | 820.0 | nM |
Neratinib | KPCD2 | 1100.0 | nM |
Neratinib | KPCD3 | 2400.0 | nM |
Neratinib | KPCE | nM | |
Neratinib | KPCI | nM | |
Neratinib | KPCL | nM | |
Neratinib | KPCT | nM | |
Neratinib | LATS1 | nM | |
Neratinib | LATS2 | nM | |
Neratinib | LCK | 120.0 | nM |
Neratinib | LIMK1 | nM | |
Neratinib | LIMK2 | nM | |
Neratinib | LKB1 | nM | |
Neratinib | LOK | 13.0 | nM |
Neratinib | LRRK2 | nM | |
Neratinib | LRRK2(G2019S) | nM | |
Neratinib | LTK | nM | |
Neratinib | LYN | 820.0 | nM |
Neratinib | M3K12 | 370.0 | nM |
Neratinib | M3K13 | 740.0 | nM |