HKI-272 KINOMEscan-2 - Dataset (ID:20195)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Neratinib | IKKB | nM | |
Neratinib | IKKE | nM | |
Neratinib | INSR | 3000.0 | nM |
Neratinib | INSRR | 4600.0 | nM |
Neratinib | IRAK1 | 2300.0 | nM |
Neratinib | IRAK3 | nM | |
Neratinib | IRAK4 | nM | |
Neratinib | ITK | nM | |
Neratinib | JAK1(JH1domain-catalytic) | nM | |
Neratinib | JAK1(JH2domain-pseudokinase) | nM | |
Neratinib | JAK2(JH1domain-catalytic) | nM | |
Neratinib | JAK3(JH1domain-catalytic) | 2000.0 | nM |
Neratinib | JNK1 | 3300.0 | nM |
Neratinib | JNK3 | 2500.0 | nM |
Neratinib | KC1G1 | nM | |
Neratinib | KC1G2 | 6600.0 | nM |
Neratinib | KCC2D | nM | |
Neratinib | KCC4 | nM | |
Neratinib | KGP1 | nM | |
Neratinib | KGP2 | nM | |
Neratinib | KIT | nM | |
Neratinib | KIT(A829P) | nM | |
Neratinib | KIT(D816H) | nM | |
Neratinib | KIT(D816V) | nM | |
Neratinib | KIT(L576P) | nM |