HKI-272 KINOMEscan-2 - Dataset (ID:20195)

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Small Molecule Protein Kd Conc unit
Neratinib MP2K2 26.0
nM
Neratinib MP2K1 14.0
nM
Neratinib MLTK 1500.0
nM
Neratinib MLK3 5800.0
nM
Neratinib MLK2 4600.0
nM
Neratinib MLK1 5400.0
nM
Neratinib MLCK
nM
Neratinib MKNK2
nM
Neratinib MKNK1
nM
Neratinib MK14
nM
Neratinib MK13
nM
Neratinib MK12
nM
Neratinib MK11
nM
Neratinib MK09
nM
Neratinib MK03
nM
Neratinib MK01
nM
Neratinib MINK 29.0
nM
Neratinib MET(Y1235D) 4200.0
nM
Neratinib MET(M1250T) 6700.0
nM
Neratinib MET 4000.0
nM
Neratinib MERTK 400.0
nM
Neratinib MELK 1600.0
nM
Neratinib MAST1 5500.0
nM
Neratinib MARK4
nM
Neratinib MARK3
nM