HKI-272 KINOMEscan-2 - Dataset (ID:20195)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Neratinib | SRPK1 | nM | |
Neratinib | SRMS | nM | |
Neratinib | SRC | 4100.0 | nM |
Neratinib | SNRK | nM | |
Neratinib | SNARK | 140.0 | nM |
Neratinib | SLK | 66.0 | nM |
Neratinib | SIK3 | nM | |
Neratinib | SIK2 | 3300.0 | nM |
Neratinib | SIK1 | 220.0 | nM |
Neratinib | SGK3 | nM | |
Neratinib | SgK110 | nM | |
Neratinib | SBK1 | nM | |
Neratinib | S6K1 | nM | |
Neratinib | RSK4(Kin.Dom.2-C-terminal) | nM | |
Neratinib | RSK4(Kin.Dom.1-N-terminal) | nM | |
Neratinib | RSK3(Kin.Dom.2-C-terminal) | nM | |
Neratinib | RSK3(Kin.Dom.1-N-terminal) | 4100.0 | nM |
Neratinib | RSK2(Kin.Dom.1-N-terminal) | nM | |
Neratinib | RSK1(Kin.Dom.2-C-terminal) | nM | |
Neratinib | RSK1(Kin.Dom.1-N-terminal) | 7400.0 | nM |
Neratinib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
Neratinib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
Neratinib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
Neratinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
Neratinib | ROS1 | nM |