HKI-272 KINOMEscan-2 - Dataset (ID:20195)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Neratinib | RSK2(Kin.Dom.1-N-terminal) | nM | |
Neratinib | RSK3(Kin.Dom.1-N-terminal) | 4100.0 | nM |
Neratinib | RSK3(Kin.Dom.2-C-terminal) | nM | |
Neratinib | RSK4(Kin.Dom.1-N-terminal) | nM | |
Neratinib | RSK4(Kin.Dom.2-C-terminal) | nM | |
Neratinib | S6K1 | nM | |
Neratinib | SBK1 | nM | |
Neratinib | SgK110 | nM | |
Neratinib | SGK3 | nM | |
Neratinib | SIK1 | 220.0 | nM |
Neratinib | SIK2 | 3300.0 | nM |
Neratinib | SLK | 66.0 | nM |
Neratinib | SNARK | 140.0 | nM |
Neratinib | SNRK | nM | |
Neratinib | SRC | 4100.0 | nM |
Neratinib | SRMS | nM | |
Neratinib | SRPK1 | nM | |
Neratinib | SRPK2 | nM | |
Neratinib | SRPK3 | nM | |
Neratinib | STK16 | nM | |
Neratinib | STK33 | 940.0 | nM |
Neratinib | STK35 | 4500.0 | nM |
Neratinib | STK36 | 5300.0 | nM |
Neratinib | STK39 | nM | |
Neratinib | SYK | 5100.0 | nM |