HKI-272 KINOMEscan-2 - Dataset (ID:20195)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Neratinib | M3K2 | 450.0 | nM |
| Neratinib | M3K5 | nM | |
| Neratinib | M3K6 | nM | |
| Neratinib | M4K1 | 93.0 | nM |
| Neratinib | M4K3 | 7.7 | nM |
| Neratinib | MAK | nM | |
| Neratinib | MAP3K1 | nM | |
| Neratinib | MAP3K15 | nM | |
| Neratinib | MAP3K3 | 130.0 | nM |
| Neratinib | MAP3K4 | 39.0 | nM |
| Neratinib | MAP4K2 | 220.0 | nM |
| Neratinib | MAP4K4 | 330.0 | nM |
| Neratinib | MAP4K5 | 0.7 | nM |
| Neratinib | MAPKAPK2 | nM | |
| Neratinib | MAPKAPK5 | nM | |
| Neratinib | MARK1 | nM | |
| Neratinib | MARK2 | nM | |
| Neratinib | MARK3 | nM | |
| Neratinib | MARK4 | nM | |
| Neratinib | MAST1 | 5500.0 | nM |
| Neratinib | MELK | 1600.0 | nM |
| Neratinib | MERTK | 400.0 | nM |
| Neratinib | MET | 4000.0 | nM |
| Neratinib | MET(M1250T) | 6700.0 | nM |
| Neratinib | MET(Y1235D) | 4200.0 | nM |