HKI-272 KINOMEscan-2 - Dataset (ID:20195)

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Small Molecule Protein Kd Conc unit
Neratinib MLTK 1500.0
nM
Neratinib NUAK1 1500.0
nM
Neratinib WEE2 1300.0
nM
Neratinib KPCD2 1100.0
nM
Neratinib DRAK2 1100.0
nM
Neratinib STK33 940.0
nM
Neratinib CHK2 850.0
nM
Neratinib KPCD1 820.0
nM
Neratinib LYN 820.0
nM
Neratinib M3K13 740.0
nM
Neratinib TNK2 680.0
nM
Neratinib CSF1R 670.0
nM
Neratinib FES 590.0
nM
Neratinib CSK 550.0
nM
Neratinib MP2K7 530.0
nM
Neratinib FER 510.0
nM
Neratinib HCK 490.0
nM
Neratinib M3K2 450.0
nM
Neratinib MERTK 400.0
nM
Neratinib TIE1 390.0
nM
Neratinib M3K12 370.0
nM
Neratinib DRAK1 340.0
nM
Neratinib MAP4K4 330.0
nM
Neratinib CSNK1E 290.0
nM
Neratinib MST1 270.0
nM