HKI-272 KINOMEscan-2 - Dataset (ID:20195)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Neratinib | INSRR | 4600.0 | nM |
| Neratinib | FLT3(D835H) | 4600.0 | nM |
| Neratinib | STK35 | 4500.0 | nM |
| Neratinib | TAOK3 | 4200.0 | nM |
| Neratinib | MET(Y1235D) | 4200.0 | nM |
| Neratinib | WEE1 | 4100.0 | nM |
| Neratinib | RSK3(Kin.Dom.1-N-terminal) | 4100.0 | nM |
| Neratinib | SRC | 4100.0 | nM |
| Neratinib | MET | 4000.0 | nM |
| Neratinib | JNK1 | 3300.0 | nM |
| Neratinib | SIK2 | 3300.0 | nM |
| Neratinib | FLT3(D835Y) | 3100.0 | nM |
| Neratinib | TIE2 | 3000.0 | nM |
| Neratinib | INSR | 3000.0 | nM |
| Neratinib | EPHB6 | 2800.0 | nM |
| Neratinib | JNK3 | 2500.0 | nM |
| Neratinib | KPCD3 | 2400.0 | nM |
| Neratinib | NEK3 | 2400.0 | nM |
| Neratinib | CDK16 | 2300.0 | nM |
| Neratinib | IRAK1 | 2300.0 | nM |
| Neratinib | JAK3(JH1domain-catalytic) | 2000.0 | nM |
| Neratinib | FGR | 1900.0 | nM |
| Neratinib | FAK1 | 1900.0 | nM |
| Neratinib | MELK | 1600.0 | nM |
| Neratinib | HIPK4 | 1500.0 | nM |