HKI-272 KINOMEscan-2 - Dataset (ID:20195)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Neratinib | FES | 590.0 | nM |
| Neratinib | FGFR1 | nM | |
| Neratinib | FGFR2 | nM | |
| Neratinib | FGFR3 | nM | |
| Neratinib | FGFR3(G697C) | nM | |
| Neratinib | FGFR4 | nM | |
| Neratinib | FGR | 1900.0 | nM |
| Neratinib | VGFR1 | nM | |
| Neratinib | FLT3 | 5400.0 | nM |
| Neratinib | FLT3(D835H) | 4600.0 | nM |
| Neratinib | FLT3(D835Y) | 3100.0 | nM |
| Neratinib | FLT3(ITD) | nM | |
| Neratinib | FLT3(K663Q) | 4900.0 | nM |
| Neratinib | FLT3(N841I) | 6400.0 | nM |
| Neratinib | FLT3(R834Q) | nM | |
| Neratinib | FLT4 | nM | |
| Neratinib | FRK | nM | |
| Neratinib | FYN | 6400.0 | nM |
| Neratinib | GAK | 250.0 | nM |
| Neratinib | GCN2(Kin.Dom.2,S808G) | 96.0 | nM |
| Neratinib | GRK1 | nM | |
| Neratinib | GRK4 | nM | |
| Neratinib | GRK7 | nM | |
| Neratinib | GSK3A | nM | |
| Neratinib | GSK3B | nM |