HKI-272 KINOMEscan-2 - Dataset (ID:20195)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Neratinib | DCAMKL2 | nM | |
| Neratinib | DCAMKL3 | nM | |
| Neratinib | DDR1 | nM | |
| Neratinib | DDR2 | nM | |
| Neratinib | M3K12 | 370.0 | nM |
| Neratinib | DMPK | nM | |
| Neratinib | DMPK2 | nM | |
| Neratinib | DRAK1 | 340.0 | nM |
| Neratinib | DRAK2 | 1100.0 | nM |
| Neratinib | DYRK1A | nM | |
| Neratinib | DYRK1B | nM | |
| Neratinib | DYRK2 | nM | |
| Neratinib | EGFR | 1.1 | nM |
| Neratinib | EGFR(E746-A750del) | 2.3 | nM |
| Neratinib | EGFR(G719C) | 0.4 | nM |
| Neratinib | EGFR(G719S) | 0.9 | nM |
| Neratinib | EGFR(L747-E749del, A750P) | 0.6 | nM |
| Neratinib | EGFR(L747-S752del, P753S) | 0.9 | nM |
| Neratinib | EGFR(L747-T751del,Sins) | 1.0 | nM |
| Neratinib | EGFR(L858R) | 0.7 | nM |
| Neratinib | EGFR(L858R,T790M) | 27.0 | nM |
| Neratinib | EGFR(L861Q) | 0.4 | nM |
| Neratinib | EGFR(S752-I759del) | 0.6 | nM |
| Neratinib | EGFR(T790M) | 1.5 | nM |
| Neratinib | EIF2AK1 | nM |