HKI-272 KINOMEscan-2 - Dataset (ID:20195)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Neratinib | MAP3K4 | 39.0 | nM |
Neratinib | MAP4K2 | 220.0 | nM |
Neratinib | M4K3 | 7.7 | nM |
Neratinib | MAP4K4 | 330.0 | nM |
Neratinib | MAP4K5 | 0.7 | nM |
Neratinib | MAPKAPK2 | nM | |
Neratinib | MAPKAPK5 | nM | |
Neratinib | MARK1 | nM | |
Neratinib | MARK2 | nM | |
Neratinib | MARK3 | nM | |
Neratinib | MARK4 | nM | |
Neratinib | MAST1 | 5500.0 | nM |
Neratinib | MP2K1 | 14.0 | nM |
Neratinib | MP2K2 | 26.0 | nM |
Neratinib | MP2K3 | nM | |
Neratinib | MP2K4 | nM | |
Neratinib | MP2K5 | 63.0 | nM |
Neratinib | MP2K6 | nM | |
Neratinib | MELK | 1600.0 | nM |
Neratinib | MERTK | 400.0 | nM |
Neratinib | MET | 4000.0 | nM |
Neratinib | MET(M1250T) | 6700.0 | nM |
Neratinib | MET(Y1235D) | 4200.0 | nM |
Neratinib | MINK | 29.0 | nM |
Neratinib | MP2K7 | 530.0 | nM |