GSK-1838705A KINOMEscan - Dataset (ID:20190)

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Small Molecule Protein Kd Conc unit
GSK1838705A ALK 0.6
nM
GSK1838705A LTK 1.1
nM
GSK1838705A INSR 1.7
nM
GSK1838705A IGF1R 7.0
nM
GSK1838705A INSRR 8.6
nM
GSK1838705A FER 9.3
nM
GSK1838705A MYLK 11.0
nM
GSK1838705A ROS1 15.0
nM
GSK1838705A CLK2 16.0
nM
GSK1838705A CLK1 21.0
nM
GSK1838705A PLK1 47.0
nM
GSK1838705A FES 52.0
nM
GSK1838705A CLK4 60.0
nM
GSK1838705A STK33 70.0
nM
GSK1838705A EGFR(T790M) 74.0
nM
GSK1838705A TTK 76.0
nM
GSK1838705A FAK2 76.0
nM
GSK1838705A JNK3 130.0
nM
GSK1838705A EGFR(L858R,T790M) 150.0
nM
GSK1838705A RSK2(Kin.Dom.1-N-terminal) 170.0
nM
GSK1838705A LRRK2(G2019S) 170.0
nM
GSK1838705A YSK4 190.0
nM
GSK1838705A FAK1 200.0
nM
GSK1838705A JNK1 210.0
nM
GSK1838705A GAK 270.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records