GSK-1838705A KINOMEscan - Dataset (ID:20190)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
GSK1838705A | ALK | 0.6 | nM |
GSK1838705A | LTK | 1.1 | nM |
GSK1838705A | INSR | 1.7 | nM |
GSK1838705A | IGF1R | 7.0 | nM |
GSK1838705A | INSRR | 8.6 | nM |
GSK1838705A | FER | 9.3 | nM |
GSK1838705A | MYLK | 11.0 | nM |
GSK1838705A | ROS1 | 15.0 | nM |
GSK1838705A | CLK2 | 16.0 | nM |
GSK1838705A | CLK1 | 21.0 | nM |
GSK1838705A | PLK1 | 47.0 | nM |
GSK1838705A | FES | 52.0 | nM |
GSK1838705A | CLK4 | 60.0 | nM |
GSK1838705A | STK33 | 70.0 | nM |
GSK1838705A | EGFR(T790M) | 74.0 | nM |
GSK1838705A | TTK | 76.0 | nM |
GSK1838705A | FAK2 | 76.0 | nM |
GSK1838705A | JNK3 | 130.0 | nM |
GSK1838705A | EGFR(L858R,T790M) | 150.0 | nM |
GSK1838705A | RSK2(Kin.Dom.1-N-terminal) | 170.0 | nM |
GSK1838705A | LRRK2(G2019S) | 170.0 | nM |
GSK1838705A | YSK4 | 190.0 | nM |
GSK1838705A | FAK1 | 200.0 | nM |
GSK1838705A | JNK1 | 210.0 | nM |
GSK1838705A | GAK | 270.0 | nM |