GSK-1838705A KINOMEscan - Dataset (ID:20190)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
GSK1838705A | IRAK1 | 8500.0 | nM |
GSK1838705A | STK16 | 7300.0 | nM |
GSK1838705A | JAK2(JH1domain-catalytic) | 5300.0 | nM |
GSK1838705A | JAK3(JH1domain-catalytic) | 4700.0 | nM |
GSK1838705A | TAK1 | 4700.0 | nM |
GSK1838705A | RIPK5 | 4300.0 | nM |
GSK1838705A | OSR1 | 4200.0 | nM |
GSK1838705A | EGFR | 4100.0 | nM |
GSK1838705A | DCLK1 | 4100.0 | nM |
GSK1838705A | EGFR(S752-I759del) | 3800.0 | nM |
GSK1838705A | CSNK1D | 3500.0 | nM |
GSK1838705A | HIPK3 | 3400.0 | nM |
GSK1838705A | TAOK1 | 3300.0 | nM |
GSK1838705A | EGFR(L747-S752del, P753S) | 3100.0 | nM |
GSK1838705A | FLT3(D835Y) | 3000.0 | nM |
GSK1838705A | RSK4(Kin.Dom.1-N-terminal) | 3000.0 | nM |
GSK1838705A | EGFR(L747-T751del,Sins) | 2900.0 | nM |
GSK1838705A | EGFR(L858R) | 2900.0 | nM |
GSK1838705A | RSK3(Kin.Dom.1-N-terminal) | 2900.0 | nM |
GSK1838705A | CSNK2A1 | 2800.0 | nM |
GSK1838705A | MERTK | 2700.0 | nM |
GSK1838705A | ERBB4 | 2400.0 | nM |
GSK1838705A | FLT3(D835H) | 2400.0 | nM |
GSK1838705A | EGFR(E746-A750del) | 2200.0 | nM |
GSK1838705A | PHKG2 | 2100.0 | nM |