GSK-1838705A KINOMEscan - Dataset (ID:20190)

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Small Molecule Protein Kd Conc unit
GSK1838705A IRAK1 8500.0
nM
GSK1838705A STK16 7300.0
nM
GSK1838705A JAK2(JH1domain-catalytic) 5300.0
nM
GSK1838705A JAK3(JH1domain-catalytic) 4700.0
nM
GSK1838705A TAK1 4700.0
nM
GSK1838705A RIPK5 4300.0
nM
GSK1838705A OSR1 4200.0
nM
GSK1838705A EGFR 4100.0
nM
GSK1838705A DCLK1 4100.0
nM
GSK1838705A EGFR(S752-I759del) 3800.0
nM
GSK1838705A CSNK1D 3500.0
nM
GSK1838705A HIPK3 3400.0
nM
GSK1838705A TAOK1 3300.0
nM
GSK1838705A EGFR(L747-S752del, P753S) 3100.0
nM
GSK1838705A FLT3(D835Y) 3000.0
nM
GSK1838705A RSK4(Kin.Dom.1-N-terminal) 3000.0
nM
GSK1838705A EGFR(L747-T751del,Sins) 2900.0
nM
GSK1838705A EGFR(L858R) 2900.0
nM
GSK1838705A RSK3(Kin.Dom.1-N-terminal) 2900.0
nM
GSK1838705A CSNK2A1 2800.0
nM
GSK1838705A MERTK 2700.0
nM
GSK1838705A ERBB4 2400.0
nM
GSK1838705A FLT3(D835H) 2400.0
nM
GSK1838705A EGFR(E746-A750del) 2200.0
nM
GSK1838705A PHKG2 2100.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records