CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | KIT | 150.0 | nM |
| Lestaurtinib | KIT(A829P) | 35.0 | nM |
| Lestaurtinib | KIT(D816H) | 11.0 | nM |
| Lestaurtinib | KIT(D816V) | 7.1 | nM |
| Lestaurtinib | KIT(L576P) | 40.0 | nM |
| Lestaurtinib | KIT(V559D) | 76.0 | nM |
| Lestaurtinib | KIT(V559D,T670I) | 45.0 | nM |
| Lestaurtinib | KIT(V559D,V654A) | 380.0 | nM |
| Lestaurtinib | LATS1 | 30.0 | nM |
| Lestaurtinib | LATS2 | 1.0 | nM |
| Lestaurtinib | LCK | 430.0 | nM |
| Lestaurtinib | LIMK1 | 1600.0 | nM |
| Lestaurtinib | LIMK2 | nM | |
| Lestaurtinib | LKB1 | 57.0 | nM |
| Lestaurtinib | LOK | 5.7 | nM |
| Lestaurtinib | LRRK2 | 3.6 | nM |
| Lestaurtinib | LRRK2(G2019S) | 2.5 | nM |
| Lestaurtinib | LTK | 490.0 | nM |
| Lestaurtinib | LYN | 190.0 | nM |
| Lestaurtinib | M3K13 | 340.0 | nM |
| Lestaurtinib | MAK | 1700.0 | nM |
| Lestaurtinib | MAP3K1 | 4400.0 | nM |
| Lestaurtinib | MAP3K15 | 3.4 | nM |
| Lestaurtinib | M3K2 | 4.8 | nM |
| Lestaurtinib | MAP3K3 | 6.0 | nM |