CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | HCK | 270.0 | nM |
| Lestaurtinib | HIPK1 | 590.0 | nM |
| Lestaurtinib | HIPK2 | 370.0 | nM |
| Lestaurtinib | HIPK3 | 250.0 | nM |
| Lestaurtinib | HIPK4 | 150.0 | nM |
| Lestaurtinib | M4K1 | 38.0 | nM |
| Lestaurtinib | HUNK | 570.0 | nM |
| Lestaurtinib | ICK | 39.0 | nM |
| Lestaurtinib | IGF1R | 4200.0 | nM |
| Lestaurtinib | IKKA | 9.0 | nM |
| Lestaurtinib | IKKB | 12.0 | nM |
| Lestaurtinib | IKKE | 11.0 | nM |
| Lestaurtinib | INSR | 1100.0 | nM |
| Lestaurtinib | INSRR | 1800.0 | nM |
| Lestaurtinib | IRAK1 | 6.1 | nM |
| Lestaurtinib | IRAK3 | 16.0 | nM |
| Lestaurtinib | IRAK4 | 1.7 | nM |
| Lestaurtinib | ITK | 290.0 | nM |
| Lestaurtinib | JAK1(JH1domain-catalytic) | 8.8 | nM |
| Lestaurtinib | JAK1(JH2domain-pseudokinase) | nM | |
| Lestaurtinib | JAK2(JH1domain-catalytic) | 3.7 | nM |
| Lestaurtinib | JAK3(JH1domain-catalytic) | 2.3 | nM |
| Lestaurtinib | JNK1 | 11.0 | nM |
| Lestaurtinib | MK09 | 320.0 | nM |
| Lestaurtinib | JNK3 | 12.0 | nM |