CEP-701 KINOMEscan - Dataset (ID:20189)

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Small Molecule Protein Kd Conc unit
Lestaurtinib ZAP70 16.0
nM
Lestaurtinib YSK4 0.5
nM
Lestaurtinib YSK1 97.0
nM
Lestaurtinib YES 160.0
nM
Lestaurtinib YANK3 8000.0
nM
Lestaurtinib YANK2 5900.0
nM
Lestaurtinib YANK1 2100.0
nM
Lestaurtinib WEE2 7900.0
nM
Lestaurtinib WEE1 1200.0
nM
Lestaurtinib VRK2
nM
Lestaurtinib VGFR2 220.0
nM
Lestaurtinib VGFR1 120.0
nM
Lestaurtinib ULK3 4.9
nM
Lestaurtinib ULK2 60.0
nM
Lestaurtinib ULK1 1000.0
nM
Lestaurtinib TYRO3 650.0
nM
Lestaurtinib TYK2(JH2domain-pseudokinase) 910.0
nM
Lestaurtinib TYK2(JH1domain-catalytic) 15.0
nM
Lestaurtinib TXK 660.0
nM
Lestaurtinib TTK 6.5
nM
Lestaurtinib TSSK1 98.0
nM
Lestaurtinib TRPM6
nM
Lestaurtinib TRKC 14.0
nM
Lestaurtinib TRKB 14.0
nM
Lestaurtinib TRKA 8.3
nM
  • Page 1 of 18
  • 1 to 25 of 442 records