CEP-701 KINOMEscan - Dataset (ID:20189)

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Small Molecule Protein Kd Conc unit
Lestaurtinib PHKG1 0.4
nM
Lestaurtinib YSK4 0.5
nM
Lestaurtinib FLT3(D835Y) 0.6
nM
Lestaurtinib FLT3(D835H) 0.7
nM
Lestaurtinib LATS2 1.0
nM
Lestaurtinib SNARK 1.0
nM
Lestaurtinib FLT3(N841I) 1.4
nM
Lestaurtinib MKNK2 1.4
nM
Lestaurtinib PLK4 1.5
nM
Lestaurtinib FLT3(ITD) 1.5
nM
Lestaurtinib IRAK4 1.7
nM
Lestaurtinib PHKG2 1.7
nM
Lestaurtinib PKN2 1.8
nM
Lestaurtinib JAK3(JH1domain-catalytic) 2.3
nM
Lestaurtinib MST2 2.4
nM
Lestaurtinib LRRK2(G2019S) 2.5
nM
Lestaurtinib CHEK1 2.8
nM
Lestaurtinib TAK1 2.9
nM
Lestaurtinib CLK4 3.0
nM
Lestaurtinib MST1 3.0
nM
Lestaurtinib AAK1 3.1
nM
Lestaurtinib DRAK1 3.4
nM
Lestaurtinib PDPK1 3.4
nM
Lestaurtinib MAP3K15 3.4
nM
Lestaurtinib MLK1 3.5
nM
  • Page 1 of 18
  • 1 to 25 of 442 records