CEP-701 KINOMEscan - Dataset (ID:20189)

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Small Molecule Protein Kd Conc unit
Lestaurtinib MK03 9800.0
nM
Lestaurtinib MRCKA 9200.0
nM
Lestaurtinib RSK4(Kin.Dom.2-C-terminal) 9100.0
nM
Lestaurtinib MST1R 8200.0
nM
Lestaurtinib OSR1 8000.0
nM
Lestaurtinib YANK3 8000.0
nM
Lestaurtinib CDK8 8000.0
nM
Lestaurtinib WEE2 7900.0
nM
Lestaurtinib ABL1(F317L)-nonphosphorylated 7600.0
nM
Lestaurtinib PIK3CA(E545K) 7400.0
nM
Lestaurtinib CSNK1A1L 7100.0
nM
Lestaurtinib EPHB2 6900.0
nM
Lestaurtinib EPHB4 6900.0
nM
Lestaurtinib PIK3CB 6700.0
nM
Lestaurtinib MLTK 6700.0
nM
Lestaurtinib RIOK2 6700.0
nM
Lestaurtinib ABL2 6500.0
nM
Lestaurtinib AKT3 6200.0
nM
Lestaurtinib YANK2 5900.0
nM
Lestaurtinib EPHA5 5900.0
nM
Lestaurtinib PIK3CA(E542K) 5900.0
nM
Lestaurtinib NEK5 5600.0
nM
Lestaurtinib PFPK5(P.falciparum) 5600.0
nM
Lestaurtinib PIK3CA(E545A) 5600.0
nM
Lestaurtinib ERBB3 5500.0
nM
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  • 1 to 25 of 442 records