SKI-606 KINOMEscan - Dataset (ID:20184)

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Small Molecule Protein Kd Conc unit
Bosutinib DCAMKL2
nM
Bosutinib DCAMKL3 5400.00
nM
Bosutinib DDR1 120.00
nM
Bosutinib DDR2 140.00
nM
Bosutinib M3K12 670.00
nM
Bosutinib DMPK 91.00
nM
Bosutinib DMPK2
nM
Bosutinib DRAK1
nM
Bosutinib DRAK2
nM
Bosutinib DYRK1A
nM
Bosutinib DYRK1B
nM
Bosutinib DYRK2
nM
Bosutinib EGFR 35.00
nM
Bosutinib EGFR(E746-A750del) 18.00
nM
Bosutinib EGFR(G719C) 98.00
nM
Bosutinib EGFR(G719S) 26.00
nM
Bosutinib EGFR(L747-E749del, A750P) 29.00
nM
Bosutinib EGFR(L747-S752del, P753S) 38.00
nM
Bosutinib EGFR(L747-T751del,Sins) 30.00
nM
Bosutinib EGFR(L858R) 23.00
nM
Bosutinib EGFR(L858R,T790M) 390.00
nM
Bosutinib EGFR(L861Q) 71.00
nM
Bosutinib EGFR(S752-I759del) 110.00
nM
Bosutinib EGFR(T790M) 340.00
nM
Bosutinib EIF2AK1 630.00
nM