SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | DCAMKL2 | nM | |
Bosutinib | DCAMKL3 | 5400.00 | nM |
Bosutinib | DDR1 | 120.00 | nM |
Bosutinib | DDR2 | 140.00 | nM |
Bosutinib | M3K12 | 670.00 | nM |
Bosutinib | DMPK | 91.00 | nM |
Bosutinib | DMPK2 | nM | |
Bosutinib | DRAK1 | nM | |
Bosutinib | DRAK2 | nM | |
Bosutinib | DYRK1A | nM | |
Bosutinib | DYRK1B | nM | |
Bosutinib | DYRK2 | nM | |
Bosutinib | EGFR | 35.00 | nM |
Bosutinib | EGFR(E746-A750del) | 18.00 | nM |
Bosutinib | EGFR(G719C) | 98.00 | nM |
Bosutinib | EGFR(G719S) | 26.00 | nM |
Bosutinib | EGFR(L747-E749del, A750P) | 29.00 | nM |
Bosutinib | EGFR(L747-S752del, P753S) | 38.00 | nM |
Bosutinib | EGFR(L747-T751del,Sins) | 30.00 | nM |
Bosutinib | EGFR(L858R) | 23.00 | nM |
Bosutinib | EGFR(L858R,T790M) | 390.00 | nM |
Bosutinib | EGFR(L861Q) | 71.00 | nM |
Bosutinib | EGFR(S752-I759del) | 110.00 | nM |
Bosutinib | EGFR(T790M) | 340.00 | nM |
Bosutinib | EIF2AK1 | 630.00 | nM |