SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | PRKX | nM | |
Bosutinib | PRP4 | nM | |
Bosutinib | FAK2 | 390.00 | nM |
Bosutinib | SIK3 | 64.00 | nM |
Bosutinib | RAF1 | nM | |
Bosutinib | RET | 4800.00 | nM |
Bosutinib | RET(M918T) | 3800.00 | nM |
Bosutinib | RET(V804L) | nM | |
Bosutinib | RET(V804M) | 4200.00 | nM |
Bosutinib | RIOK1 | 2200.00 | nM |
Bosutinib | RIOK2 | nM | |
Bosutinib | RIOK3 | 1600.00 | nM |
Bosutinib | RIPK1 | nM | |
Bosutinib | RIPK2 | 3700.00 | nM |
Bosutinib | RIPK4 | nM | |
Bosutinib | RIPK5 | 380.00 | nM |
Bosutinib | ROCK1 | 870.00 | nM |
Bosutinib | ROCK2 | 360.00 | nM |
Bosutinib | ROS1 | nM | |
Bosutinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
Bosutinib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
Bosutinib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
Bosutinib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
Bosutinib | RSK1(Kin.Dom.1-N-terminal) | nM | |
Bosutinib | RSK1(Kin.Dom.2-C-terminal) | nM |