SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | MET(M1250T) | 6800.00 | nM |
Bosutinib | TYK2(JH1domain-catalytic) | 6500.00 | nM |
Bosutinib | MST1R | 6300.00 | nM |
Bosutinib | MYO3A | 6200.00 | nM |
Bosutinib | NUAK1 | 5900.00 | nM |
Bosutinib | CTK | 5800.00 | nM |
Bosutinib | PAK3 | 5700.00 | nM |
Bosutinib | PKNB(M.tuberculosis) | 5500.00 | nM |
Bosutinib | DCAMKL3 | 5400.00 | nM |
Bosutinib | MP2K7 | 5300.00 | nM |
Bosutinib | PGFRA | 5100.00 | nM |
Bosutinib | HUNK | 5000.00 | nM |
Bosutinib | GRK4 | 4900.00 | nM |
Bosutinib | RET | 4800.00 | nM |
Bosutinib | TSSK1 | 4600.00 | nM |
Bosutinib | KPCD3 | 4600.00 | nM |
Bosutinib | TYK2(JH2domain-pseudokinase) | 4500.00 | nM |
Bosutinib | CAMK2A | 4500.00 | nM |
Bosutinib | MAP3K1 | 4400.00 | nM |
Bosutinib | RET(V804M) | 4200.00 | nM |
Bosutinib | SRPK3 | 3900.00 | nM |
Bosutinib | AMPK-alpha1 | 3900.00 | nM |
Bosutinib | TIE2 | 3900.00 | nM |
Bosutinib | RET(M918T) | 3800.00 | nM |
Bosutinib | STK39 | 3700.00 | nM |