BMS-540215 KINOMEscan - Dataset (ID:20180)

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Small Molecule Protein Kd Conc unit
Brivanib ABL1(T315I)-phosphorylated 450.0
nM
Brivanib ABL1(M351T)-phosphorylated 450.0
nM
Brivanib YSK4 500.0
nM
Brivanib ABL1(E255K)-phosphorylated 580.0
nM
Brivanib MAP4K4 590.0
nM
Brivanib FGFR4 600.0
nM
Brivanib ABL1-phosphorylated 640.0
nM
Brivanib ABL1(H396P)-phosphorylated 640.0
nM
Brivanib ABL1-nonphosphorylated 1100.0
nM
Brivanib ABL1(Y253F)-phosphorylated 1100.0
nM
Brivanib LCK 1100.0
nM
Brivanib TIE1 1100.0
nM
Brivanib ABL1(Q252H)-phosphorylated 1200.0
nM
Brivanib MAP4K5 1400.0
nM
Brivanib EPHB6 1400.0
nM
Brivanib ABL1(Q252H)-nonphosphorylated 1500.0
nM
Brivanib SRC 1600.0
nM
Brivanib ABL1(T315I)-nonphosphorylated 1700.0
nM
Brivanib EPHA7 1700.0
nM
Brivanib ABL2 1800.0
nM
Brivanib CSF1R 1900.0
nM
Brivanib BLK 2000.0
nM
Brivanib ABL1(F317L)-phosphorylated 2300.0
nM
Brivanib EGFR(G719S) 2600.0
nM
Brivanib HCK 2700.0
nM