BMS-540215 KINOMEscan - Dataset (ID:20180)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Brivanib | ABL1(T315I)-phosphorylated | 450.0 | nM |
Brivanib | ABL1(M351T)-phosphorylated | 450.0 | nM |
Brivanib | YSK4 | 500.0 | nM |
Brivanib | ABL1(E255K)-phosphorylated | 580.0 | nM |
Brivanib | MAP4K4 | 590.0 | nM |
Brivanib | FGFR4 | 600.0 | nM |
Brivanib | ABL1-phosphorylated | 640.0 | nM |
Brivanib | ABL1(H396P)-phosphorylated | 640.0 | nM |
Brivanib | ABL1-nonphosphorylated | 1100.0 | nM |
Brivanib | ABL1(Y253F)-phosphorylated | 1100.0 | nM |
Brivanib | LCK | 1100.0 | nM |
Brivanib | TIE1 | 1100.0 | nM |
Brivanib | ABL1(Q252H)-phosphorylated | 1200.0 | nM |
Brivanib | MAP4K5 | 1400.0 | nM |
Brivanib | EPHB6 | 1400.0 | nM |
Brivanib | ABL1(Q252H)-nonphosphorylated | 1500.0 | nM |
Brivanib | SRC | 1600.0 | nM |
Brivanib | ABL1(T315I)-nonphosphorylated | 1700.0 | nM |
Brivanib | EPHA7 | 1700.0 | nM |
Brivanib | ABL2 | 1800.0 | nM |
Brivanib | CSF1R | 1900.0 | nM |
Brivanib | BLK | 2000.0 | nM |
Brivanib | ABL1(F317L)-phosphorylated | 2300.0 | nM |
Brivanib | EGFR(G719S) | 2600.0 | nM |
Brivanib | HCK | 2700.0 | nM |