Sunitinib KINOMEscan - Dataset (ID:20179)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Sunitinib | PRKX | nM | |
Sunitinib | PRP4 | 390.0 | nM |
Sunitinib | FAK2 | 82.0 | nM |
Sunitinib | SIK3 | nM | |
Sunitinib | RAF1 | nM | |
Sunitinib | RET | 13.0 | nM |
Sunitinib | RET(M918T) | 19.0 | nM |
Sunitinib | RET(V804L) | 8.7 | nM |
Sunitinib | RET(V804M) | 5.8 | nM |
Sunitinib | RIOK1 | 35.0 | nM |
Sunitinib | RIOK2 | 49.0 | nM |
Sunitinib | RIOK3 | 3800.0 | nM |
Sunitinib | RIPK1 | 370.0 | nM |
Sunitinib | RIPK2 | nM | |
Sunitinib | RIPK4 | 2100.0 | nM |
Sunitinib | RIPK5 | 1300.0 | nM |
Sunitinib | ROCK1 | 460.0 | nM |
Sunitinib | ROCK2 | 140.0 | nM |
Sunitinib | ROS1 | nM | |
Sunitinib | RPS6KA4(Kin.Dom.1-N-terminal) | 96.0 | nM |
Sunitinib | RPS6KA4(Kin.Dom.2-C-terminal) | 2000.0 | nM |
Sunitinib | RPS6KA5(Kin.Dom.1-N-terminal) | 28.0 | nM |
Sunitinib | RPS6KA5(Kin.Dom.2-C-terminal) | 1700.0 | nM |
Sunitinib | RSK1(Kin.Dom.1-N-terminal) | 140.0 | nM |
Sunitinib | RSK1(Kin.Dom.2-C-terminal) | 5000.0 | nM |