Sunitinib KINOMEscan - Dataset (ID:20179)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Sunitinib | IKKB | nM | |
Sunitinib | IKKE | 620.0 | nM |
Sunitinib | INSR | 500.0 | nM |
Sunitinib | INSRR | 430.0 | nM |
Sunitinib | IRAK1 | 14.0 | nM |
Sunitinib | IRAK3 | 940.0 | nM |
Sunitinib | IRAK4 | 66.0 | nM |
Sunitinib | ITK | 13.0 | nM |
Sunitinib | JAK1(JH1domain-catalytic) | 6000.0 | nM |
Sunitinib | JAK1(JH2domain-pseudokinase) | 49.0 | nM |
Sunitinib | JAK2(JH1domain-catalytic) | 410.0 | nM |
Sunitinib | JAK3(JH1domain-catalytic) | 1200.0 | nM |
Sunitinib | JNK1 | nM | |
Sunitinib | JNK3 | 4300.0 | nM |
Sunitinib | KC1G1 | 930.0 | nM |
Sunitinib | KC1G2 | 110.0 | nM |
Sunitinib | KCC2D | 420.0 | nM |
Sunitinib | KCC4 | 890.0 | nM |
Sunitinib | KGP1 | nM | |
Sunitinib | KGP2 | nM | |
Sunitinib | KIT | 0.4 | nM |
Sunitinib | KIT(A829P) | 43.0 | nM |
Sunitinib | KIT(D816H) | 110.0 | nM |
Sunitinib | KIT(D816V) | 380.0 | nM |
Sunitinib | KIT(L576P) | 1.3 | nM |