Sunitinib KINOMEscan - Dataset (ID:20179)

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Small Molecule Protein Kd Conc unit
Sunitinib IKKB
nM
Sunitinib IKKE 620.0
nM
Sunitinib INSR 500.0
nM
Sunitinib INSRR 430.0
nM
Sunitinib IRAK1 14.0
nM
Sunitinib IRAK3 940.0
nM
Sunitinib IRAK4 66.0
nM
Sunitinib ITK 13.0
nM
Sunitinib JAK1(JH1domain-catalytic) 6000.0
nM
Sunitinib JAK1(JH2domain-pseudokinase) 49.0
nM
Sunitinib JAK2(JH1domain-catalytic) 410.0
nM
Sunitinib JAK3(JH1domain-catalytic) 1200.0
nM
Sunitinib JNK1
nM
Sunitinib JNK3 4300.0
nM
Sunitinib KC1G1 930.0
nM
Sunitinib KC1G2 110.0
nM
Sunitinib KCC2D 420.0
nM
Sunitinib KCC4 890.0
nM
Sunitinib KGP1
nM
Sunitinib KGP2
nM
Sunitinib KIT 0.4
nM
Sunitinib KIT(A829P) 43.0
nM
Sunitinib KIT(D816H) 110.0
nM
Sunitinib KIT(D816V) 380.0
nM
Sunitinib KIT(L576P) 1.3
nM