Sunitinib KINOMEscan - Dataset (ID:20179)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Sunitinib | PGFRB | 0.1 | nM |
| Sunitinib | FLT3(K663Q) | 0.2 | nM |
| Sunitinib | KIT(V559D,V654A) | 0.2 | nM |
| Sunitinib | KIT(V559D,T670I) | 0.3 | nM |
| Sunitinib | KIT | 0.4 | nM |
| Sunitinib | KIT(V559D) | 0.4 | nM |
| Sunitinib | FLT3 | 0.4 | nM |
| Sunitinib | PGFRA | 0.8 | nM |
| Sunitinib | DRAK1 | 1.0 | nM |
| Sunitinib | FLT3(ITD) | 1.0 | nM |
| Sunitinib | KIT(L576P) | 1.3 | nM |
| Sunitinib | VGFR2 | 1.5 | nM |
| Sunitinib | VGFR1 | 1.8 | nM |
| Sunitinib | FLT3(D835Y) | 2.3 | nM |
| Sunitinib | FLT3(N841I) | 2.4 | nM |
| Sunitinib | CSF1R | 2.5 | nM |
| Sunitinib | FLT3(D835H) | 4.3 | nM |
| Sunitinib | BIKE | 5.5 | nM |
| Sunitinib | PHKG1 | 5.5 | nM |
| Sunitinib | RET(V804M) | 5.8 | nM |
| Sunitinib | PHKG2 | 5.9 | nM |
| Sunitinib | RET(V804L) | 8.7 | nM |
| Sunitinib | AXL | 9.0 | nM |
| Sunitinib | CHK2 | 10.0 | nM |
| Sunitinib | FLT3(R834Q) | 11.0 | nM |