Sunitinib KINOMEscan - Dataset (ID:20179)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Sunitinib | FES | 960.0 | nM |
Sunitinib | FGFR1 | 520.0 | nM |
Sunitinib | FGFR2 | 570.0 | nM |
Sunitinib | FGFR3 | 290.0 | nM |
Sunitinib | FGFR3(G697C) | 1400.0 | nM |
Sunitinib | FGFR4 | 2100.0 | nM |
Sunitinib | FGR | 270.0 | nM |
Sunitinib | VGFR1 | 1.8 | nM |
Sunitinib | FLT3 | 0.4 | nM |
Sunitinib | FLT3(D835H) | 4.3 | nM |
Sunitinib | FLT3(D835Y) | 2.3 | nM |
Sunitinib | FLT3(ITD) | 1.0 | nM |
Sunitinib | FLT3(K663Q) | 0.2 | nM |
Sunitinib | FLT3(N841I) | 2.4 | nM |
Sunitinib | FLT3(R834Q) | 11.0 | nM |
Sunitinib | FLT4 | 50.0 | nM |
Sunitinib | FRK | 530.0 | nM |
Sunitinib | FYN | 520.0 | nM |
Sunitinib | GAK | 20.0 | nM |
Sunitinib | GCN2(Kin.Dom.2,S808G) | 180.0 | nM |
Sunitinib | GRK1 | 290.0 | nM |
Sunitinib | GRK4 | 140.0 | nM |
Sunitinib | GRK7 | 180.0 | nM |
Sunitinib | GSK3A | nM | |
Sunitinib | GSK3B | nM |