Sunitinib KINOMEscan - Dataset (ID:20179)

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Small Molecule Protein Kd Conc unit
Sunitinib FES 960.0
nM
Sunitinib FGFR1 520.0
nM
Sunitinib FGFR2 570.0
nM
Sunitinib FGFR3 290.0
nM
Sunitinib FGFR3(G697C) 1400.0
nM
Sunitinib FGFR4 2100.0
nM
Sunitinib FGR 270.0
nM
Sunitinib VGFR1 1.8
nM
Sunitinib FLT3 0.4
nM
Sunitinib FLT3(D835H) 4.3
nM
Sunitinib FLT3(D835Y) 2.3
nM
Sunitinib FLT3(ITD) 1.0
nM
Sunitinib FLT3(K663Q) 0.2
nM
Sunitinib FLT3(N841I) 2.4
nM
Sunitinib FLT3(R834Q) 11.0
nM
Sunitinib FLT4 50.0
nM
Sunitinib FRK 530.0
nM
Sunitinib FYN 520.0
nM
Sunitinib GAK 20.0
nM
Sunitinib GCN2(Kin.Dom.2,S808G) 180.0
nM
Sunitinib GRK1 290.0
nM
Sunitinib GRK4 140.0
nM
Sunitinib GRK7 180.0
nM
Sunitinib GSK3A
nM
Sunitinib GSK3B
nM