Sunitinib KINOMEscan - Dataset (ID:20179)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Sunitinib | DCAMKL2 | 2700.0 | nM |
Sunitinib | DCAMKL3 | 110.0 | nM |
Sunitinib | DDR1 | 2000.0 | nM |
Sunitinib | DDR2 | 2900.0 | nM |
Sunitinib | M3K12 | 100.0 | nM |
Sunitinib | DMPK | nM | |
Sunitinib | DMPK2 | nM | |
Sunitinib | DRAK1 | 1.0 | nM |
Sunitinib | DRAK2 | 110.0 | nM |
Sunitinib | DYRK1A | 200.0 | nM |
Sunitinib | DYRK1B | 2300.0 | nM |
Sunitinib | DYRK2 | 680.0 | nM |
Sunitinib | EGFR | nM | |
Sunitinib | EGFR(E746-A750del) | nM | |
Sunitinib | EGFR(G719C) | 6800.0 | nM |
Sunitinib | EGFR(G719S) | nM | |
Sunitinib | EGFR(L747-E749del, A750P) | nM | |
Sunitinib | EGFR(L747-S752del, P753S) | nM | |
Sunitinib | EGFR(L747-T751del,Sins) | nM | |
Sunitinib | EGFR(L858R) | nM | |
Sunitinib | EGFR(L858R,T790M) | 860.0 | nM |
Sunitinib | EGFR(L861Q) | nM | |
Sunitinib | EGFR(S752-I759del) | nM | |
Sunitinib | EGFR(T790M) | 2400.0 | nM |
Sunitinib | EIF2AK1 | nM |