GSK-1363089 KINOMEscan - Dataset (ID:20176)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Foretinib | KIT | 2.5 | nM |
| Foretinib | KIT(A829P) | 3.2 | nM |
| Foretinib | KIT(D816H) | 36.0 | nM |
| Foretinib | KIT(D816V) | 9.6 | nM |
| Foretinib | KIT(L576P) | 2.7 | nM |
| Foretinib | KIT(V559D) | 2.1 | nM |
| Foretinib | KIT(V559D,T670I) | 2.4 | nM |
| Foretinib | KIT(V559D,V654A) | 7.6 | nM |
| Foretinib | LATS1 | nM | |
| Foretinib | LATS2 | nM | |
| Foretinib | LCK | 6.0 | nM |
| Foretinib | LIMK1 | 680.0 | nM |
| Foretinib | LIMK2 | 1700.0 | nM |
| Foretinib | LKB1 | nM | |
| Foretinib | LOK | 0.5 | nM |
| Foretinib | LRRK2 | nM | |
| Foretinib | LRRK2(G2019S) | nM | |
| Foretinib | LTK | 110.0 | nM |
| Foretinib | LYN | 9.1 | nM |
| Foretinib | M3K13 | 16.0 | nM |
| Foretinib | MAK | 1800.0 | nM |
| Foretinib | MAP3K1 | nM | |
| Foretinib | MAP3K15 | nM | |
| Foretinib | M3K2 | 1900.0 | nM |
| Foretinib | MAP3K3 | 4800.0 | nM |