GSK-1363089 KINOMEscan - Dataset (ID:20176)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Foretinib | HCK | 15.0 | nM |
Foretinib | HIPK1 | 420.0 | nM |
Foretinib | HIPK2 | 220.0 | nM |
Foretinib | HIPK3 | 43.0 | nM |
Foretinib | HIPK4 | 0.5 | nM |
Foretinib | M4K1 | 44.0 | nM |
Foretinib | HUNK | 5400.0 | nM |
Foretinib | ICK | nM | |
Foretinib | IGF1R | 430.0 | nM |
Foretinib | IKKA | 5900.0 | nM |
Foretinib | IKKB | nM | |
Foretinib | IKKE | 1400.0 | nM |
Foretinib | INSR | 210.0 | nM |
Foretinib | INSRR | 53.0 | nM |
Foretinib | IRAK1 | nM | |
Foretinib | IRAK3 | 370.0 | nM |
Foretinib | IRAK4 | nM | |
Foretinib | ITK | 69.0 | nM |
Foretinib | JAK1(JH1domain-catalytic) | nM | |
Foretinib | JAK1(JH2domain-pseudokinase) | nM | |
Foretinib | JAK2(JH1domain-catalytic) | 1500.0 | nM |
Foretinib | JAK3(JH1domain-catalytic) | nM | |
Foretinib | JNK1 | 5700.0 | nM |
Foretinib | MK09 | 670.0 | nM |
Foretinib | JNK3 | 3900.0 | nM |