GSK-1363089 KINOMEscan - Dataset (ID:20176)

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Small Molecule Protein Kd Conc unit
Foretinib HCK 15.0
nM
Foretinib HIPK1 420.0
nM
Foretinib HIPK2 220.0
nM
Foretinib HIPK3 43.0
nM
Foretinib HIPK4 0.5
nM
Foretinib M4K1 44.0
nM
Foretinib HUNK 5400.0
nM
Foretinib ICK
nM
Foretinib IGF1R 430.0
nM
Foretinib IKKA 5900.0
nM
Foretinib IKKB
nM
Foretinib IKKE 1400.0
nM
Foretinib INSR 210.0
nM
Foretinib INSRR 53.0
nM
Foretinib IRAK1
nM
Foretinib IRAK3 370.0
nM
Foretinib IRAK4
nM
Foretinib ITK 69.0
nM
Foretinib JAK1(JH1domain-catalytic)
nM
Foretinib JAK1(JH2domain-pseudokinase)
nM
Foretinib JAK2(JH1domain-catalytic) 1500.0
nM
Foretinib JAK3(JH1domain-catalytic)
nM
Foretinib JNK1 5700.0
nM
Foretinib MK09 670.0
nM
Foretinib JNK3 3900.0
nM