TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib CAMK1G 3200.0
nM
Fedratinib TESK1 3200.0
nM
Fedratinib MLK1 3200.0
nM
Fedratinib EGFR(L858R) 3300.0
nM
Fedratinib EGFR 3400.0
nM
Fedratinib NEK1 3400.0
nM
Fedratinib MP2K3 3500.0
nM
Fedratinib KIT(V559D,V654A) 3500.0
nM
Fedratinib ZAP70 3800.0
nM
Fedratinib CHEK1 3800.0
nM
Fedratinib KGP1 3800.0
nM
Fedratinib PAK4 3800.0
nM
Fedratinib EGFR(L747-T751del,Sins) 3800.0
nM
Fedratinib EPHB2 3900.0
nM
Fedratinib EPHA6 3900.0
nM
Fedratinib PIK3CA(H1047L) 3900.0
nM
Fedratinib EPHA4 4000.0
nM
Fedratinib CAMKK2 4000.0
nM
Fedratinib MAP3K4 4100.0
nM
Fedratinib PI42C 4100.0
nM
Fedratinib ANKK1 4300.0
nM
Fedratinib VGFR1 4300.0
nM
Fedratinib AURKA 4400.0
nM
Fedratinib RPS6KA5(Kin.Dom.1-N-terminal) 4400.0
nM
Fedratinib MET(M1250T) 4400.0
nM