TG-101348 KINOMEscan - Dataset (ID:20174)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Fedratinib | FES | 530.0 | nM |
| Fedratinib | FGFR1 | 280.0 | nM |
| Fedratinib | FGFR2 | 470.0 | nM |
| Fedratinib | FGFR3 | 360.0 | nM |
| Fedratinib | FGFR3(G697C) | 760.0 | nM |
| Fedratinib | FGFR4 | 2000.0 | nM |
| Fedratinib | FGR | 82.0 | nM |
| Fedratinib | VGFR1 | 4300.0 | nM |
| Fedratinib | FLT3 | 13.0 | nM |
| Fedratinib | FLT3(D835H) | 4.9 | nM |
| Fedratinib | FLT3(D835Y) | 6.4 | nM |
| Fedratinib | FLT3(ITD) | 16.0 | nM |
| Fedratinib | FLT3(K663Q) | 13.0 | nM |
| Fedratinib | FLT3(N841I) | 20.0 | nM |
| Fedratinib | FLT3(R834Q) | 29.0 | nM |
| Fedratinib | FLT4 | 2000.0 | nM |
| Fedratinib | FRK | 200.0 | nM |
| Fedratinib | FYN | 38.0 | nM |
| Fedratinib | GAK | 1.1 | nM |
| Fedratinib | GCN2(Kin.Dom.2,S808G) | 100.0 | nM |
| Fedratinib | GRK1 | nM | |
| Fedratinib | GRK4 | 170.0 | nM |
| Fedratinib | GRK7 | 2600.0 | nM |
| Fedratinib | GSK3A | nM | |
| Fedratinib | GSK3B | nM |