TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib M3K2 580.0
nM
Fedratinib M3K5
nM
Fedratinib M3K6
nM
Fedratinib M4K1 1300.0
nM
Fedratinib M4K3 1800.0
nM
Fedratinib MAK
nM
Fedratinib MAP3K1
nM
Fedratinib MAP3K15
nM
Fedratinib MAP3K3 1300.0
nM
Fedratinib MAP3K4 4100.0
nM
Fedratinib MAP4K2 2100.0
nM
Fedratinib MAP4K4
nM
Fedratinib MAP4K5
nM
Fedratinib MAPKAPK2
nM
Fedratinib MAPKAPK5
nM
Fedratinib MARK1 700.0
nM
Fedratinib MARK2 3100.0
nM
Fedratinib MARK3 300.0
nM
Fedratinib MARK4 970.0
nM
Fedratinib MAST1
nM
Fedratinib MELK 2600.0
nM
Fedratinib MERTK 820.0
nM
Fedratinib MET 8500.0
nM
Fedratinib MET(M1250T) 4400.0
nM
Fedratinib MET(Y1235D)
nM