TG-101348 KINOMEscan - Dataset (ID:20174)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | M3K2 | 580.0 | nM |
Fedratinib | M3K5 | nM | |
Fedratinib | M3K6 | nM | |
Fedratinib | M4K1 | 1300.0 | nM |
Fedratinib | M4K3 | 1800.0 | nM |
Fedratinib | MAK | nM | |
Fedratinib | MAP3K1 | nM | |
Fedratinib | MAP3K15 | nM | |
Fedratinib | MAP3K3 | 1300.0 | nM |
Fedratinib | MAP3K4 | 4100.0 | nM |
Fedratinib | MAP4K2 | 2100.0 | nM |
Fedratinib | MAP4K4 | nM | |
Fedratinib | MAP4K5 | nM | |
Fedratinib | MAPKAPK2 | nM | |
Fedratinib | MAPKAPK5 | nM | |
Fedratinib | MARK1 | 700.0 | nM |
Fedratinib | MARK2 | 3100.0 | nM |
Fedratinib | MARK3 | 300.0 | nM |
Fedratinib | MARK4 | 970.0 | nM |
Fedratinib | MAST1 | nM | |
Fedratinib | MELK | 2600.0 | nM |
Fedratinib | MERTK | 820.0 | nM |
Fedratinib | MET | 8500.0 | nM |
Fedratinib | MET(M1250T) | 4400.0 | nM |
Fedratinib | MET(Y1235D) | nM |