TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib PKNB(M.tuberculosis) 100.0
nM
Fedratinib GCN2(Kin.Dom.2,S808G) 100.0
nM
Fedratinib SRPK2 100.0
nM
Fedratinib RIOK1 100.0
nM
Fedratinib ABL1(Q252H)-nonphosphorylated 110.0
nM
Fedratinib NEK6 120.0
nM
Fedratinib CSNK2A2 120.0
nM
Fedratinib IRAK3 120.0
nM
Fedratinib YES 120.0
nM
Fedratinib CDK7 120.0
nM
Fedratinib KIT(L576P) 120.0
nM
Fedratinib MYLK4 130.0
nM
Fedratinib RET 130.0
nM
Fedratinib KIT 130.0
nM
Fedratinib RPS6KA4(Kin.Dom.2-C-terminal) 140.0
nM
Fedratinib CIT 140.0
nM
Fedratinib RET(M918T) 150.0
nM
Fedratinib NEK9 150.0
nM
Fedratinib ACVR1 150.0
nM
Fedratinib KIT(D816H) 160.0
nM
Fedratinib KIT(D816V) 160.0
nM
Fedratinib NEK7 160.0
nM
Fedratinib SRPK1 160.0
nM
Fedratinib PIP5K2B 160.0
nM
Fedratinib AXL 160.0
nM