TG-101348 KINOMEscan - Dataset (ID:20174)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | PKNB(M.tuberculosis) | 100.0 | nM |
Fedratinib | GCN2(Kin.Dom.2,S808G) | 100.0 | nM |
Fedratinib | SRPK2 | 100.0 | nM |
Fedratinib | RIOK1 | 100.0 | nM |
Fedratinib | ABL1(Q252H)-nonphosphorylated | 110.0 | nM |
Fedratinib | NEK6 | 120.0 | nM |
Fedratinib | CSNK2A2 | 120.0 | nM |
Fedratinib | IRAK3 | 120.0 | nM |
Fedratinib | YES | 120.0 | nM |
Fedratinib | CDK7 | 120.0 | nM |
Fedratinib | KIT(L576P) | 120.0 | nM |
Fedratinib | MYLK4 | 130.0 | nM |
Fedratinib | RET | 130.0 | nM |
Fedratinib | KIT | 130.0 | nM |
Fedratinib | RPS6KA4(Kin.Dom.2-C-terminal) | 140.0 | nM |
Fedratinib | CIT | 140.0 | nM |
Fedratinib | RET(M918T) | 150.0 | nM |
Fedratinib | NEK9 | 150.0 | nM |
Fedratinib | ACVR1 | 150.0 | nM |
Fedratinib | KIT(D816H) | 160.0 | nM |
Fedratinib | KIT(D816V) | 160.0 | nM |
Fedratinib | NEK7 | 160.0 | nM |
Fedratinib | SRPK1 | 160.0 | nM |
Fedratinib | PIP5K2B | 160.0 | nM |
Fedratinib | AXL | 160.0 | nM |