TG-101348 KINOMEscan - Dataset (ID:20174)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | ABL1(H396P)-nonphosphorylated | 45.0 | nM |
Fedratinib | PGFRB | 45.0 | nM |
Fedratinib | DRAK2 | 45.0 | nM |
Fedratinib | KIT(A829P) | 46.0 | nM |
Fedratinib | SNARK | 49.0 | nM |
Fedratinib | ABL1(M351T)-phosphorylated | 50.0 | nM |
Fedratinib | ABL1(Q252H)-phosphorylated | 54.0 | nM |
Fedratinib | ABL1(Y253F)-phosphorylated | 56.0 | nM |
Fedratinib | KIT(V559D) | 58.0 | nM |
Fedratinib | ABL1(H396P)-phosphorylated | 61.0 | nM |
Fedratinib | TNK2 | 64.0 | nM |
Fedratinib | ABL1(T315I)-phosphorylated | 65.0 | nM |
Fedratinib | PIP5K1A | 66.0 | nM |
Fedratinib | ERK5 | 66.0 | nM |
Fedratinib | RET(V804L) | 71.0 | nM |
Fedratinib | LCK | 72.0 | nM |
Fedratinib | JAK3(JH1domain-catalytic) | 74.0 | nM |
Fedratinib | SRC | 75.0 | nM |
Fedratinib | ULK2 | 79.0 | nM |
Fedratinib | RET(V804M) | 81.0 | nM |
Fedratinib | FGR | 82.0 | nM |
Fedratinib | RIOK3 | 91.0 | nM |
Fedratinib | TBK1 | 92.0 | nM |
Fedratinib | PLK4 | 96.0 | nM |
Fedratinib | SIK2 | 98.0 | nM |