TG-101348 KINOMEscan - Dataset (ID:20174)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | BRAF | 9800.0 | nM |
Fedratinib | BMX | 1200.0 | nM |
Fedratinib | BMPR2 | 2900.0 | nM |
Fedratinib | BMPR1B | 410.0 | nM |
Fedratinib | BMPR1A | nM | |
Fedratinib | BLK | 650.0 | nM |
Fedratinib | BIKE | 32.0 | nM |
Fedratinib | AXL | 160.0 | nM |
Fedratinib | AURKC | 350.0 | nM |
Fedratinib | AURKB | 490.0 | nM |
Fedratinib | AURKA | 4400.0 | nM |
Fedratinib | ANKK1 | 4300.0 | nM |
Fedratinib | AMPK-alpha2 | 4700.0 | nM |
Fedratinib | AMPK-alpha1 | 2400.0 | nM |
Fedratinib | ALK | 650.0 | nM |
Fedratinib | AKT3 | nM | |
Fedratinib | AKT2 | nM | |
Fedratinib | AKT1 | nM | |
Fedratinib | ADCK4 | 300.0 | nM |
Fedratinib | ADCK3 | 7000.0 | nM |
Fedratinib | ACVRL1 | 2400.0 | nM |
Fedratinib | ACVR2B | nM | |
Fedratinib | ACVR2A | nM | |
Fedratinib | ACVR1B | 6700.0 | nM |
Fedratinib | ACVR1 | 150.0 | nM |