TG-101348 KINOMEscan - Dataset (ID:20174)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | LIMK2 | 7900.0 | nM |
Fedratinib | LIMK1 | 940.0 | nM |
Fedratinib | LCK | 72.0 | nM |
Fedratinib | LATS2 | 8000.0 | nM |
Fedratinib | LATS1 | nM | |
Fedratinib | KPCT | nM | |
Fedratinib | KPCL | nM | |
Fedratinib | KPCI | nM | |
Fedratinib | KPCE | 8100.0 | nM |
Fedratinib | KPCD3 | 9600.0 | nM |
Fedratinib | KPCD2 | nM | |
Fedratinib | KPCD1 | nM | |
Fedratinib | KPCD | nM | |
Fedratinib | KKCC1 | 1800.0 | nM |
Fedratinib | KIT(V559D,V654A) | 3500.0 | nM |
Fedratinib | KIT(V559D,T670I) | 1500.0 | nM |
Fedratinib | KIT(V559D) | 58.0 | nM |
Fedratinib | KIT(L576P) | 120.0 | nM |
Fedratinib | KIT(D816V) | 160.0 | nM |
Fedratinib | KIT(D816H) | 160.0 | nM |
Fedratinib | KIT(A829P) | 46.0 | nM |
Fedratinib | KIT | 130.0 | nM |
Fedratinib | KGP2 | 1600.0 | nM |
Fedratinib | KGP1 | 3800.0 | nM |
Fedratinib | KCC4 | nM |