TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib LIMK2 7900.0
nM
Fedratinib LIMK1 940.0
nM
Fedratinib LCK 72.0
nM
Fedratinib LATS2 8000.0
nM
Fedratinib LATS1
nM
Fedratinib KPCT
nM
Fedratinib KPCL
nM
Fedratinib KPCI
nM
Fedratinib KPCE 8100.0
nM
Fedratinib KPCD3 9600.0
nM
Fedratinib KPCD2
nM
Fedratinib KPCD1
nM
Fedratinib KPCD
nM
Fedratinib KKCC1 1800.0
nM
Fedratinib KIT(V559D,V654A) 3500.0
nM
Fedratinib KIT(V559D,T670I) 1500.0
nM
Fedratinib KIT(V559D) 58.0
nM
Fedratinib KIT(L576P) 120.0
nM
Fedratinib KIT(D816V) 160.0
nM
Fedratinib KIT(D816H) 160.0
nM
Fedratinib KIT(A829P) 46.0
nM
Fedratinib KIT 130.0
nM
Fedratinib KGP2 1600.0
nM
Fedratinib KGP1 3800.0
nM
Fedratinib KCC4
nM