TG-101348 KINOMEscan - Dataset (ID:20174)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | ZAP70 | 3800.0 | nM |
Fedratinib | YSK4 | 19.0 | nM |
Fedratinib | YSK1 | 7200.0 | nM |
Fedratinib | YES | 120.0 | nM |
Fedratinib | YANK3 | nM | |
Fedratinib | YANK2 | nM | |
Fedratinib | YANK1 | nM | |
Fedratinib | WEE2 | 6000.0 | nM |
Fedratinib | WEE1 | 390.0 | nM |
Fedratinib | VRK2 | nM | |
Fedratinib | VGFR2 | 5200.0 | nM |
Fedratinib | VGFR1 | 4300.0 | nM |
Fedratinib | ULK3 | 290.0 | nM |
Fedratinib | ULK2 | 79.0 | nM |
Fedratinib | ULK1 | 270.0 | nM |
Fedratinib | TYRO3 | nM | |
Fedratinib | TYK2(JH2domain-pseudokinase) | 450.0 | nM |
Fedratinib | TYK2(JH1domain-catalytic) | 21.0 | nM |
Fedratinib | TXK | 1500.0 | nM |
Fedratinib | TTK | 450.0 | nM |
Fedratinib | TSSK1 | 1300.0 | nM |
Fedratinib | TRPM6 | nM | |
Fedratinib | TRKC | 8600.0 | nM |
Fedratinib | TRKB | 3100.0 | nM |
Fedratinib | TRKA | 840.0 | nM |