TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib MLK2 6900.0
nM
Fedratinib PAK6 6900.0
nM
Fedratinib CAMK2B 6800.0
nM
Fedratinib ACVR1B 6700.0
nM
Fedratinib EPHA7 6500.0
nM
Fedratinib LTK 6300.0
nM
Fedratinib M3K12 6300.0
nM
Fedratinib EGFR(E746-A750del) 6200.0
nM
Fedratinib RIPK2 6100.0
nM
Fedratinib PAK2 6000.0
nM
Fedratinib WEE2 6000.0
nM
Fedratinib CSK 5900.0
nM
Fedratinib NDR1 5800.0
nM
Fedratinib EGFR(L861Q) 5800.0
nM
Fedratinib EGFR(L747-S752del, P753S) 5600.0
nM
Fedratinib RIPK1 5300.0
nM
Fedratinib VGFR2 5200.0
nM
Fedratinib MP2K1 5100.0
nM
Fedratinib SRMS 5000.0
nM
Fedratinib CDK4-cyclinD1 5000.0
nM
Fedratinib AMPK-alpha2 4700.0
nM
Fedratinib RPS6KA5(Kin.Dom.1-N-terminal) 4400.0
nM
Fedratinib NIM1 4400.0
nM
Fedratinib EPHA2 4400.0
nM
Fedratinib AURKA 4400.0
nM