TG-101348 KINOMEscan - Dataset (ID:20174)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | MLK2 | 6900.0 | nM |
Fedratinib | PAK6 | 6900.0 | nM |
Fedratinib | CAMK2B | 6800.0 | nM |
Fedratinib | ACVR1B | 6700.0 | nM |
Fedratinib | EPHA7 | 6500.0 | nM |
Fedratinib | LTK | 6300.0 | nM |
Fedratinib | M3K12 | 6300.0 | nM |
Fedratinib | EGFR(E746-A750del) | 6200.0 | nM |
Fedratinib | RIPK2 | 6100.0 | nM |
Fedratinib | PAK2 | 6000.0 | nM |
Fedratinib | WEE2 | 6000.0 | nM |
Fedratinib | CSK | 5900.0 | nM |
Fedratinib | NDR1 | 5800.0 | nM |
Fedratinib | EGFR(L861Q) | 5800.0 | nM |
Fedratinib | EGFR(L747-S752del, P753S) | 5600.0 | nM |
Fedratinib | RIPK1 | 5300.0 | nM |
Fedratinib | VGFR2 | 5200.0 | nM |
Fedratinib | MP2K1 | 5100.0 | nM |
Fedratinib | SRMS | 5000.0 | nM |
Fedratinib | CDK4-cyclinD1 | 5000.0 | nM |
Fedratinib | AMPK-alpha2 | 4700.0 | nM |
Fedratinib | RPS6KA5(Kin.Dom.1-N-terminal) | 4400.0 | nM |
Fedratinib | NIM1 | 4400.0 | nM |
Fedratinib | EPHA2 | 4400.0 | nM |
Fedratinib | AURKA | 4400.0 | nM |