TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib PIP5K1A 66.0
nM
Fedratinib PIP5K1C
nM
Fedratinib PIP5K2B 160.0
nM
Fedratinib PI42C 4100.0
nM
Fedratinib PKAC-alpha
nM
Fedratinib PKAC-beta
nM
Fedratinib PKMYT1
nM
Fedratinib PKN1 1100.0
nM
Fedratinib PKN2
nM
Fedratinib PKNB(M.tuberculosis) 100.0
nM
Fedratinib PLK1 280.0
nM
Fedratinib PLK2 2400.0
nM
Fedratinib PLK3 1600.0
nM
Fedratinib PLK4 96.0
nM
Fedratinib KPCD
nM
Fedratinib KPCE 8100.0
nM
Fedratinib KPCL
nM
Fedratinib KPCI
nM
Fedratinib KPCT
nM
Fedratinib KPCD1
nM
Fedratinib KPCD2
nM
Fedratinib KPCD3 9600.0
nM
Fedratinib KGP1 3800.0
nM
Fedratinib KGP2 1600.0
nM
Fedratinib PRKR 1100.0
nM