INCB018424 KINOMEscan - Dataset (ID:20173)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Ruxolitinib | FES | nM | |
Ruxolitinib | FGFR1 | nM | |
Ruxolitinib | FGFR2 | nM | |
Ruxolitinib | FGFR3 | nM | |
Ruxolitinib | FGFR3(G697C) | nM | |
Ruxolitinib | FGFR4 | nM | |
Ruxolitinib | FGR | nM | |
Ruxolitinib | VGFR1 | nM | |
Ruxolitinib | FLT3 | nM | |
Ruxolitinib | FLT3(D835H) | nM | |
Ruxolitinib | FLT3(D835Y) | nM | |
Ruxolitinib | FLT3(ITD) | nM | |
Ruxolitinib | FLT3(K663Q) | nM | |
Ruxolitinib | FLT3(N841I) | nM | |
Ruxolitinib | FLT3(R834Q) | nM | |
Ruxolitinib | FLT4 | nM | |
Ruxolitinib | FRK | nM | |
Ruxolitinib | FYN | nM | |
Ruxolitinib | GAK | 99.0 | nM |
Ruxolitinib | GCN2(Kin.Dom.2,S808G) | nM | |
Ruxolitinib | GRK1 | 730.0 | nM |
Ruxolitinib | GRK4 | 6100.0 | nM |
Ruxolitinib | GRK7 | 540.0 | nM |
Ruxolitinib | GSK3A | nM | |
Ruxolitinib | GSK3B | nM |